Prosecution Insights
Last updated: April 17, 2026
Application No. 18/126,250

DNA-ENCODED AND AFFINITY-TAGGED MASKED-WARHEAD COMPOUNDS AND USE THEREOF IN ASSEMBLING LIBRARIES OF SMALL MOLECULES ENABLED FOR LATE-STAGE PURIFICATION AND MULTIPLEXED SCREENING OF COVALENT LIGANDS

Non-Final OA §102
Filed
Mar 24, 2023
Examiner
FLINDERS, JEREMY C
Art Unit
1684
Tech Center
1600 — Biotechnology & Organic Chemistry
Assignee
unknown
OA Round
1 (Non-Final)
64%
Grant Probability
Moderate
1-2
OA Rounds
3y 9m
To Grant
80%
With Interview

Examiner Intelligence

Grants 64% of resolved cases
64%
Career Allow Rate
378 granted / 586 resolved
+4.5% vs TC avg
Strong +15% interview lift
Without
With
+15.2%
Interview Lift
resolved cases with interview
Typical timeline
3y 9m
Avg Prosecution
48 currently pending
Career history
634
Total Applications
across all art units

Statute-Specific Performance

§101
8.8%
-31.2% vs TC avg
§103
33.2%
-6.8% vs TC avg
§102
26.1%
-13.9% vs TC avg
§112
21.1%
-18.9% vs TC avg
Black line = Tech Center average estimate • Based on career data from 586 resolved cases

Office Action

§102
DETAILED ACTION Status of the Claims Claims 1-15 are currently pending and are the subject of this Office Action. The present application, filed on or after March 16, 2013, is being examined under the first inventor to file provisions of the AIA . Information Disclosure Statement The information disclosure statement (IDS) submitted on 07/28/2023 is in compliance with the provisions of 37 CFR 1.97. Accordingly, the information disclosure statement is being considered by the examiner. Claim Objections Claims 2 and 14 are objected to as being dependent upon rejected base claims, but would be free from the prior art if rewritten in independent form including all of the limitations of the base claims and any intervening claims. Appropriate correction is required. Claim Rejections – 35 U.S.C. 102 In the event the determination of the status of the application as subject to AIA 35 U.S.C. 102 and 103 (or as subject to pre-AIA 35 U.S.C. 102 and 103) is incorrect, any correction of the statutory basis for the rejection will not be considered a new ground of rejection if the prior art relied upon, and the rationale supporting the rejection, would be the same under either status. The following is a quotation of the appropriate paragraphs of 35 U.S.C. 102 that form the basis for the rejections under this section made in this Office action: A person shall be entitled to a patent unless – (a)(1) the claimed invention was patented, described in a printed publication, or in public use, on sale or otherwise available to the public before the effective filing date of the claimed invention. (a)(2) the claimed invention was described in a patent issued under section 151, or in an application for patent published or deemed published under section 122(b), in which the patent or application, as the case may be, names another inventor and was effectively filed before the effective filing date of the claimed invention. Faucher et al. Claim 1 is rejected under 35 U.S.C. 102(a)(1) as being anticipated by Faucher et al. (J. Med. Chem., 2004, 47:18-21). Regarding claim 1, Faucher discloses a compound represented by formula (I): PNG media_image1.png 120 414 media_image1.png Greyscale , for example, those in the right column of Table 1, wherein (B) is a phenyl group with Y=Y1=CH with R3’=H, (Linker) is a covalent bond, affinity tag (A) is covalently bound to the phenyl group varies among Entries 14-25, n=0, and R2’ and R2’’ are each H. Newlander et al. Claims 12-13 are rejected under 35 U.S.C. 102(a)(1) as being anticipated by Newlander et al. (J. Org. Chem., 1997, 62:6726-6732). Regarding claims 12-13, Newlander discloses a compound represented by formula (II): PNG media_image2.png 126 424 media_image2.png Greyscale for example, compound 24 on p. 6728, wherein (B) is a phenyl group with Y=Y1=CH with R3’=H, (Linker) is a covalent bond, affinity tag (A) is PNG media_image3.png 82 140 media_image3.png Greyscale covalently bound to the phenyl group, n=1, R1’=R1’’=R2’=R2’’=H, and R4’=R4’’=CH3. Wang et al. Claims 3-11 and 15 are rejected under 35 U.S.C. 102(a)(1) as being anticipated by Wang et al. (Org. Lett., 2019, 21:719−723). Claims 3 and 15 recite eDELs, which are generated from the methods of claims 2 and 14, respectively, and are therefore product-by-process claims. Note that as per MPEP § 2113, “product-by-process claims are not limited to the manipulations of the recited steps, only the structure implied by the steps”. The same MPEP section states that “‘even though product-by-process claims are limited by and defined by the process, determination of patentability is based on the product itself. The patentability of a product does not depend on its method of production. If the product in the product-by-process claim is the same as or obvious from a product of the prior art, the claim is unpatentable even though the prior product was made by a different process.’ In re Thorpe, 777 F.2d 695, 698, 227 USPQ 964, 966 (Fed. Cir. 1985). In the present case, the process steps imply the structural limitations as shown in, for example, Fig. 2B-2: PNG media_image4.png 200 232 media_image4.png Greyscale Wang teaches several acrylamide-type structures that are encompassed by this formula, such as those listed in Tables 1 and 2, and these products meets all of the structural limitations of the claimed product (see above) except for the product-by-process limitations and thus would either anticipate or render obvious the claimed composition comprising activated eDELs set forth in claims 3 and 15. Here, Applicants’ claims are drawn to activated eDELs (i.e., products), but are defined by various method steps that produce said eDELs (e.g. coupling formula I or II with a DEL to generate a mwDEL, purifying the mwDEL intermediate, unmasking the mwDEL to generate an activate eDEL, and purifying the activated eDEL) and, as a result, represent product-by-process claims. Thus, the specific process limitations of claims 2 and 14 do not distinguish the claimed invention from the prior art in accordance with MPEP § 2113. One of ordinary skill would expect the product to be the same no matter how it was synthesized and/or prepared. Alternatively or in addition, a plurality of structures in Fig. 1A of the present disclosure represent eDELs from the prior art which could have reasonably been made by the methods of claims 2 and/or 14, thus anticipating the eDELs of claims 3 and 15. For example, Fig. 1A-4 could reasonably be made, wherein R1=CH3 and R2=H: PNG media_image5.png 188 168 media_image5.png Greyscale Conclusion No claims are allowed. Any inquiry concerning this communication or earlier communications from the examiner should be directed to JEREMY FLINDERS whose telephone number is (571)270-1022. The examiner can normally be reached M-F 10-6:00 EST. Examiner interviews are available via telephone, in-person, and video conferencing using a USPTO supplied web-based collaboration tool. To schedule an interview, applicant is encouraged to use the USPTO Automated Interview Request (AIR) at http://www.uspto.gov/interviewpractice. If attempts to reach the examiner by telephone are unsuccessful, the examiner’s supervisor, Heather Calamita can be reached on (571)272-2876. The fax phone number for the organization where this application or proceeding is assigned is 571-273-8300. Information regarding the status of published or unpublished applications may be obtained from Patent Center. Unpublished application information in Patent Center is available to registered users. To file and manage patent submissions in Patent Center, visit: https://patentcenter.uspto.gov. Visit https://www.uspto.gov/patents/apply/patent-center for more information about Patent Center and https://www.uspto.gov/patents/docx for information about filing in DOCX format. For additional questions, contact the Electronic Business Center (EBC) at 866-217-9197 (toll-free). If you would like assistance from a USPTO Customer Service Representative, call 800-786-9199 (IN USA OR CANADA) or 571-272-1000. /JEREMY C FLINDERS/ Primary Examiner, Art Unit 1684
Read full office action

Prosecution Timeline

Mar 24, 2023
Application Filed
Jan 27, 2026
Non-Final Rejection — §102 (current)

Precedent Cases

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Study what changed to get past this examiner. Based on 5 most recent grants.

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Prosecution Projections

1-2
Expected OA Rounds
64%
Grant Probability
80%
With Interview (+15.2%)
3y 9m
Median Time to Grant
Low
PTA Risk
Based on 586 resolved cases by this examiner. Grant probability derived from career allow rate.

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